HYDRATE OF 1-{(2S)}2-AMINO-4-[2,4-BIS(TRIFLUOROMETHYL)-5,8-DI-HYDROPYRIDO[3,4-d]PYRIMIDIN-7(6H)-YL]-4-OXOBUTYL}-5,5-DIFLUORO-PIPERIDIN-2-ONE TARTRATE
关于老挝专利「HYDRATE OF 1-{(2S)}2-AMINO-4-[2,4-BIS(TRIFLUOROMETHYL)-5,8-DI-HYDROPYRIDO[3,4-d]PYRIMIDIN-7(6H)-YL]-4-OXOBUTYL}-5,5-DIFLUORO-PIPERIDIN-2-ONE TARTRATE」,老商通整理了如下公开信息,由 LG CHEM, LTD. 于 2011-10-27 提交申请,当前状态为已注册。公开档案中可核验:申请号 P/161,DIP 编号 LAP161,主管局代码 LA,保护类型 Patent - Foreign。时间线要点:公开/公告日 2022-10-07;授权日 2022-10-04;届满/失效参考日 2031-10-27。国际分类 / IPC 标注为 C07D 471/04。发明人 / 设计人包括 KIM, Bong Chan、KIM, Kyu Young、LEE, Ji Hye、PARK, Ki Sook、YUN, Jung Min。代理机构 / 代理人记载为 Lao Trademark Agency。公开摘要提示:The present invention relates to 1.5 hydrate of 1-{(2S)-2-amino-4-[2,4-bis(trifluoromethyl)-5,8-dihydropyrido[3,4-d]pyrimidin-7(6H)-yl]-4-o…。
LaoBiz profiles the Laos patent “HYDRATE OF 1-{(2S)}2-AMINO-4-[2,4-BIS(TRIFLUOROMETHYL)-5,8-DI-HYDROPYRIDO[3,4-d]PYRIMIDIN-7(6H)-YL]-4-OXOBUTYL}-5,5-DIFLUORO-PIPERIDIN-2-ONE TARTRATE” from open registry fields, filed by LG CHEM, LTD. on 2011-10-27; current status: Registered. Identifiers include application No. P/161; DIP id LAP161; protection kind Patent - Foreign. Key dates: publication 2022-10-07; grant 2022-10-04; expiry reference 2031-10-27. Classification: C07D 471/04. Inventor(s)/designer(s): KIM, Bong Chan, KIM, Kyu Young, LEE, Ji Hye, PARK, Ki Sook, YUN, Jung Min. Abstract hint: The present invention relates to 1.5 hydrate of 1-{(2S)-2-amino-4-[2,4-bis(trifluoromethyl)-5,8-dihydropyrido[3,4-d]pyrimidin-7(6H)-yl]-4-o…. This prose is informational only and does not constitute legal advice, ownership proof or an infringement opinion.
ສິດທິບັດ «HYDRATE OF 1-{(2S)}2-AMINO-4-[2,4-BIS(TRIFLUOROMETHYL)-5,8-DI-HYDROPYRIDO[3,4-d]PYRIMIDIN-7(6H)-YL]-4-OXOBUTYL}-5,5-DIFLUORO-PIPERIDIN-2-ONE TARTRATE» ເປັນຂໍ້ມູນຊັບສິນທາງປັນຍາເປີດເຜີຍຂອງ DIP, ຍື່ນໂດຍ LG CHEM, LTD. ໃນວັນທີ 2011-10-27; ສະຖານະ ຈົດທະບຽນແລ້ວ. ຕົວລະບຸ: ເລກທີຄຳຮ້ອງ P/161; ລະຫັດ DIP LAP161; ປະເພດການປົກປ້ອງ Patent - Foreign. ວັນທີສຳຄັນ: ວັນເຜີຍແຜ່ 2022-10-07; ວັນຈົດທະບຽນ/ອະນຸຍາດ 2022-10-04; ວັນໝົດອາຍຸ 2031-10-27. ປະເພດ/ຫ້ອງ: C07D 471/04. ນັກປະດິດ/ນັກອອກແບບ: KIM, Bong Chan, KIM, Kyu Young, LEE, Ji Hye, PARK, Ki Sook, YUN, Jung Min. ສະຫຼຸບ: ສິ່ງຄົ້ນຄິດນີ້- ພົວພັນເຖິງ 1.5 ໄຮເດຣທ໌ ຂອງ 1-{(2S)-2-ອາມີໂນ-4-[2,4-ບິສ(ໄຕຣຟລູອໍໂຣເມທິລ)-5,8-ໄດໄຣໂດຣເພີໄຣໂດ [3,4-d]ເພີຣີມີດີນ-7(6H)--yl]-4-ອ…. ຂໍ້ມູນເພື່ອອ້າງອີງເທົ່ານັ້ນ ບໍ່ແມ່ນຄຳແນະນຳທາງກົດໝາຍ ຫຼື ໃບຢັ້ງຢືນສິດ.
P/161
图样
基础信息
- 类型
- 专利
- 申请号
P/161- 状态
- 已注册
- 申请人
- LG CHEM, LTD.
- 代理机构
- Lao Trademark Agency
- 申请日期
- 2011-10-27
- 注册号
P/161- 公开/公告日
- 2022-10-07
- 注册/授权日
- 2022-10-04
- 届满日
- 2031-10-27
- 国际分类
- C07D 471/04
- 商品 / 服务
- —
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摘要
ສິ່ງຄົ້ນຄິດນີ້- ພົວພັນເຖິງ 1.5 ໄຮເດຣທ໌ ຂອງ 1-{(2S)-2-ອາມີໂນ-4-[2,4-ບິສ(ໄຕຣຟລູອໍໂຣເມທິລ)-5,8-ໄດໄຣໂດຣເພີໄຣໂດ [3,4-d]ເພີຣີມີດີນ-7(6H)--yl]-4-ອອັກໂຊບິວທິລ}-5,5-ໄຕຣຟລູອໍໂຣໄພເພີຣີດີນ -2-ວັນ ທາເທຣດທ໌, ຂະບວນການສຳລັບກນປຸງແຕ່ງອັນດຽວກັນ, ແລະ ສ່ວນປະກອບ ທາງການຢາ ສຳລັບການຢັບຢັ້ງ DPP-IV, ຊື່ງ ປະກອບດ້ວຍສານປະກອບທີ່ວ່ານັ້ນເປັນສານປະກອບທີ່ແຂງແຮງ
The present invention relates to 1.5 hydrate of 1-{(2S)-2-amino-4-[2,4-bis(trifluoromethyl)-5,8-dihydropyrido[3,4-d]pyrimidin-7(6H)-yl]-4-oxobutyl}-5,5-difluoropiperidin-2-one tartrate, a process for preparing the same, and a pharmaceutical composition for inhibiting DPP-IV, which comprises said compound as the active component.